Publications 201

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Poreba M, Groborz K, Navarro M, Snipas SJ, Drag M, Salvesen GS, Caspase selective reagents for diagnosing apoptotic mechanisms Cell Death and Differentiation 2019, 26, 229.

Burda‐Grabowska, M.; Macegoniuk, K.; Flick, R.; Nocek, B. P.; Joachimiak, A.; Yakunin, A. F.; Mucha, A.; Berlicki, Ł., Bisphosphonic acids and related compounds as inhibitors of nucleotide‐ and polyphosphate‐processing enzymes: A PPK1 and PPK2 case study. Chem. Biol. Drug Des. 2019, 93, 1197.

Cogo F, Poreba M, Rut W, Groborz K, Smyth P, Johnston MC, Williams R, Longley DB, Burden RE, Salvesen GS, Drag M, Scott Ch., Development of an advanced nanoformulation for the intracellular delivery of a caspase-3 selective activity-based probe Nanoscale 2019, 11, 742.

Strub, D.J., Szymanska, K., Hrydziuszko, Z., Bryjak, J., Jarzebski, A.B., Continuous flow kinetic resolution of a non-equimolar mixture of diastereoisomeric alcohol using a structured monolithic enzymatic microreactor React. Chem. Eng. 2019, 4, 587.

Hrydziuszko, Z., Strub, D., Labus, K., Bryjak, J., Burkholderia cepacia lipase immobilization for hydrolytic reactions and the kinetic resolution of the non-equimolar mixtures of isomeric alcohols Bioorg Chem 2019, accepted.

Kozioł, A., Jasnowski, M., Grela, E., Szczepanik, M., Gabryś, B., Dancewicz, K., Lochyński, S.,, Synthesis and Biological Activity of New 4‐tert‐Butylcyclohexanone Derivatives Chem. Biodiversity 2019, 16, 1.

Kozioł, A., Grela, E., Macegoniuk, K.M., Grabowiecka, A., Lochyński, S., Synthesis of nitrogen-containing monoterpenoids with antibacterial activity Nat. Prod. Res., 2019, 1.

Vallade M., Jewgiński M., Fischer L., Buratto J., Bathany K., Schmitter J.M., Stupfel M., Godde F., Mackereth C.D., Huc I., Assessing Interactions between Helical Aromatic Oligoamide Foldamers and Protein Surfaces: A Tethering Approach Bioconjugate Chemistry 2019, 30, 54.

Stanek, N.; Teper, D.; Kafarski, P.; Jasicka-Misiak, I., Authentication of phacelia honeys (Phacelia tanacetifolia) based on a combination of HPLC and HPTLC analyses as well as spectrophotometric measurements LWT - Food Science and Technology 2019, 107, 199.

Pagoni, A.; Daliani, T.; Macegoniuk, K.; Vassiliou, S.; Berlicki, Ł., Catechol-based inhibitors of bacterial urease Bioorg. Med. Chem. Lett. 2019, 29, 1085.

Katarzyna Hałdys, Rafał Latajka, Thiosemicarbazones with tyrosinase inhibitory activity MedChemComm 2019, 10, 378.

Talma, M.; Maślanka, M.; Mucha, A., Recent developments in the synthesis and applications of phosphinic peptide analogs. Bioorg. Med. Chem. Lett. 2019, 29, 1031.

Bak, A., Kozik V., Kozakiewicz D., Gajcy K., Strub D.J., Swietlicka A., Stepankova S., Imramovsky A., Polanski J, Smolinski A., Jampilek, J., Novel Benzene-based Carbamates for AChE/BChE Inhibition: Synthesis and Ligand/Structure-oriented SAR study Int. J. Mol. Sci. 2019, 20, 1.

Schröder D.C., Kracker O., Fröhr T., Góra J., Jewginski M., Nieß A., Antes I., Latajka R., Marion A., Sewald N., 1,4-Disubstituted 1H-1,2,3-Triazole Containing Peptidotriazolamers: A New Class of Peptidomimetics With Interesting Foldamer Properties Frontiers in Chemistry 2019, 7, 1.

Poreba M, Rut W, Groborz K, Snipas SJ, Salvesen GS, Drag M, Potent and selective caspase-2 inhibitor prevents MDM-2 cleavage in reversine-treated colon cancer cells Cell Death and Differentiation 2019, 26, 2695.

Poreba M, Recent advances in the development of legumain-selective chemical probes and peptide prodrugs Biological Chemistry 2019, 1.

Groborz K, Kolt S, Kasperkiewicz P, Drag M, Internally Quenched Fluorogenic substrates with unnatural amino acids for cathepsin G investigation Biochimie 2019, 166, 103.

Argüello-Velasco, R. O.; Dziuk, B.; Zarychta, B.; Ordóñez, M.; Kafarski, P., Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin- 3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations ACS Omega 2019, 4, 9056.

Stanek, N,; Kafarski, P.; Jasicka-Misiak, I., Development of a high performance thin layer chromatography method for the rapid qualification and quantification of phenolic compounds and abscisic acid in honeys J. Chromatogr. A 2019, 1598, 209.

Wolinska, E.; Hałdys, K.; Góra, J.; Olszewski, T.K.; Boduszek, B.; Latajka, R., Phosphonic and phosphinic acid derivatives as novel tyrosinaseinhibitors: Kinetic studies and molecular docking. Chem. Biodiversity 2019, 1.

de Vries LE, Sanchez MI, Groborz K, Kuppens L, Poreba M, Lehmann C, Nevins N, Withers-Martinez C, Hirst DJ, Yuan F, Arastu-Kapur S, Horn M, Mares M, Bogyo M, Drag M, Deu E, Characterization of P. falciparum dipeptidyl aminopeptidase 3 specificity identifies differences in amino acid preferences between peptide-based substrates and covalent inhibitors FEBS Journal 2019, 286, 3998.

Groborz K, Gonzalez-Ramirez ML, Snipas SJ, Salvesen GS, Drag M, Poreba M, Exploring the prime site in caspases as a novel chemical strategy for understanding the mechanisms of cell death: a proof of concept study on necroptosis in cancer cells Cell Death and Differentiation 2019, 1.

Maślanka, M.; Mucha, A., Recent Developments in Peptidyl Diaryl Phoshonates as Inhibitors and Activity-Based Probes for Serine Proteases Pharmaceuticals 2019, 12, 86.

Drąg-Zalesińska M, Rembiałkowska N, Borska S, Saczko J, Drąg M, Poręba M, Kulbacka J, A New Betulin Derivative Stimulates the Synthesis of Collagen in Human Fibroblasts Stronger than its Precursor In vivo 2019, 33, 1087.

Argüello-Velasco, R. O.; Sánchez-Muñoz, K. O.; Viveros-Ceballos, J. L.; Ordóñez, M.; Kafarski, P., A Straightforward Synthesis of Six-Membered-Ring Heterocyclic α-Aminophosphonic Acids from N-Acyliminium Ions J. Heterocyclic Chem. 2019, 56, 2068.

Balcerzak, L., Gibka, J., Sikora, M., Kula, J., Strub, D.J., Minor constituents of essential oils and aromatic extracts. Oximes derived from natural flavor and fragrance raw materials - sensory evaluation, spectral and gas chromatographic characteristics Food Chemistry 2019, accepted.

Poreba M, Groborz K, Vizovisek M, Maruggi M, Turk D, Turk B, Powis G, Drag M, Salvesen GS, Fluorescent probes towards selective cathepsin B detection and visualization in cancer cells and patient samples Chemical Science 2019, 10, 8461.

Rut W, Nielsen NV, Czarna J, Poreba M, Kanse SM, Drag M, Fluorescent activity-based probe for the selective detection of Factor VII activating protease (FSAP) in human plasma Thrombosis Research 2019, 182, 124.

Babin BM, Kasperkiewicz P, Janiszewski T, Yoo E, Drag M, Bogyo M, Leveraging peptide substrate libraries to design inhibitors of bacterial Lon protease ACS Chemical Biology 2019, 1.

Urbańczyk M., Jewgiński M, Krzciuk-Gula J., Góra J., Latajka R., Sewald N., Synthesis and conformational preferences of short analogues of antifreeze glycopeptides (AFGP) Beilstein J. Org. Chem. 2019, 15, 1581.

Makowicz, E.; Jasicka-Misiak, I.; Teper, D.; Kafarski, P., Botanical Origin Authentication of Polish Phacelia Honey Using the Combination of Volatile Fraction Profiling by HS‑SPME and Lipophilic Fraction Profiling by HPTLC Chromatographia 2019, 82, 1541.

Wanat, W.; Talma, M.; Pawełczak, M.; Kafarski, P., Phosphonic Acid Analogues of Phenylglycine as Inhibitors of Aminopeptidases: Comparison of Porcine Aminopeptidase N, Bovine Leucine Aminopeptidase, Tomato Acidic Leucine Aminopeptidase and Aminopeptidase from Barley Seeds Pharmaceuticals 2019, 12, 1.

Anderson BM, Poole DP, Aurelio L, Ng GZ, Fleischmann M, Kasperkiewicz P, Morissette C, Drag M, van Driel IR, Schmidt BL, Vanner SJ, Bunnett NW, Edgington-Mitchell LE, Application of a chemical probe to detect neutrophil elastase activation during inflammatory bowel disease Scientific Reports 2019, 9, 13295.

Poreba M, Groborz K, Rut W, Pore M, Snipas SJ, Vizovisek M, Turk B, Drag M, Salvesen GS, The Activome: multiplexed probing of activity of proteolytic enzymes using mass cytometry-compatible activity-based probes (TOF-probes) bioRxiv 2019, 1.

Aaltonen N, Singha P, Jakupovic H, Wirth T, Samaranayake H, Pasonen-Seppanen S, Rilla K, Varjosalo M, Edgington-Mitchell L, Kasperkiewicz P, Drag M, Kalvala S, Moisio E, Savinainen JR, Laitinen JT, Tissue-ABPP enables high-resolution confocal fluorescence imaging of serine hydrolase activity in cryosections – Application to glioma brain unveils activity hotspots originating from tumor-associated neutrophils bioRxiv 2019, 1.

Maluch I, Czarna J, Drag M, Applications of unnatural amino acids in protease probes Chemistry - An Asian Journal 2019, 14, 4103.

Ignatiuk, Z. A.; Janicki, M. J.; Gora, R. W.; Konieczny, K.; Kowalczyk, R. , Applications of Thermal Activation, Ball-milling and Aqueous Medium in Stereoselective Michael Addition of Nitromethane to Enynones Catalyzed by Chiral Squaramides Advanced Synthesis & Catalysis 2019, 361, 1108.

Lunde NN, Gregersen I, Ueland T, Shetelig C, Holm S, Kong XY, Michelsen AE, Otterdal K, Yndestad A, Broch K, Gullestad L, Nyman TA, Bendz B, Eritsland J, Hoffmann P, Skagen K, Gonçalves I, Nilsson J, Grenegård M, Poreba M, Drag M, Seljeflot I, Sporsheim B, Espevik T, Skjelland M, Johansen HT, Solberg R, Aukrust P, Björkbacka H, Andersen GØ, Halvorsen B, Legumain is upregulated in acute cardiovascular events and associated with improved outcome - potentially related to anti-inflammatory effects on macrophages. Atherosclerosis 2019, 1.

Stosiek, N.; Talma, M.; Klimek-Ochab, M., Carbon-Phosphorus Lyase—the State of the Art Appl. Biochem. Biotechnol. 2019, 1.