Publications 2016

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Kosikowska, P.; Bochno, M.; Macegoniuk, K.; Forlani, G.; Kafarski, P.; Berlicki, Ł., Bisphosphonic acids as effective inhibitors of Mycobacterium tuberculosis glutamine synthetase J. Enz. Inh. Med. Chem. 2016, 31, 931.

Wójcik, P.; Berlicki, Ł., Peptide-based inhibitors of protein–protein interactions. Bioorg. Med. Chem. Lett. 2016, 26, 707.

Górny vel Górniak, M.; Kafarski, P., Preparation of the library of fluorescent aromatic aminophosphonate phenyl and benzyl esters Phosphorus, Sulfur, Silicon Relat. Elem. 2016, 191, 511.

Węglarz-Tomczak, E.; Berlicki, Ł.; Pawełczak, M.; Nocek, B.; Joachimiak, A. Mucha, A., A structural insight into the P1-S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases. Eur. J. Med. Chem. 2016, 117, 187.

Chmielewska, E.; Kafarski, P., Physiologic Activity of Bisphosphonates – Recent Advances Open Pharm. Sci. J. 2016, 3, 56.

Dziuganowska, Z. A.; Ślepokura, A.; Volle, J.-N.; Virieux, D.; Pirat, J.-L.; Kafarski, P., Structural Analogues of Selfotel J. Org. Chem. 2016, 81, 4947.

Macegoniuk, K.; Grela, E.; Palus, J.; Rudzińska-Szostak, E.; Grabowiecka, A.; Biernat, M.; Berlicki, Ł., 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. J. Med. Chem. 2016, 59, 8125.

Węglarz-Tomczak, E.; Vassiliou, S.; Mucha, A., Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues. Bioorg. Med. Chem. Lett. 2016, 26, 4122.

Węglarz-Tomczak, E.; Staszewska, K.; Talma, M.; Mucha, A., Enantiomeric a,ß-diaminoethylphosphonic acids as potent inhibitors of aminopeptidases — stereoselective synthesis and biological activity. Tetrahedron Lett. 2016, 57, 4812.

Węglarz-Tomczak, E.; Burda-Grabowska, M.; Giurg, M.; Mucha, A., Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study. Bioorg. Med. Chem. Lett. 2016, 26, 5254.

Grela, E.; Dziełak, A.; Szydowska, K.; Mucha, A.; Kafarski, P.; Grabowiecka, A.M., Whole-cell Proteus mirabilis urease inhibition by aminophosphinates for the control of struvite formation. J. Med. Microbiol. 2016, 65, 1123.

Chmielewska, E.; Kafarski, P., Synthetic procedures leading towards aminobisphosphonates Molecules 2016, 21, 1.

Dobosz, A.; Spychała, J.; Ptak, T.; Chmielewska, E.; Maciejewska, G.; Kafarski, P.; Młynarz, P. , Electrochemical and spectroscopic investigations of selected N-heteroalkylaminomethylenebisphosphonic acids with Pb(II) ions Coord. Chem. Rev. 2016, 327-328, 271.

Jewginski, M., Fischer, L., Colombo, C., Huc, I., MacKereth, C.D., Solution Observation of Dimerization and Helix Handedness Induction in a Human Carbonic Anhydrase-Helical Aromatic Amide Foldamer Complex ChemBioChem 2016, 17, 727.

Lamch, Ł.; Tylus, W.; Jewgiński, M.; Latajka, R.; Wilk, K.A., Location of Varying Hydrophobicity Zinc(II) Phthalocyanine-Type Photosensitizers in Methoxy Poly(ethylene oxide) and Poly(L‑lactide) Block Copolymer Micelles Using 1H NMR and XPS Techniques. J. Phys. Chem. B 2016, 120, 12768.

Boratynski, P.J. ; Kowalczyk, R., Click-Dimerized Cinchona Alkaloids JOURNAL OF ORGANIC CHEMISTRY 2016, 81, 8029.

Boratynski, P.J.; Kowalczyk, R.; Kobylanska, A.; Bakowicz, J., Tricyclic Quaternary Ammonium Salts Derived from Cinchona Alkaloids JOURNAL OF ORGANIC CHEMISTRY 2016, 81, 12489.

Kowalczyk, R.; Boratynski, P.J. , Stereoselective thia-Michael 1,4-Addition to Acyclic 2,4-Dienones and 2-En-4-ynones ADVANCED SYNTHESIS & CATALYSIS 2016, 358, 1289.

Rebelo, S. L. H.; Guedes, A.; Szefczyk, M. E.; Pereira, A. M.; Araujo, J. P.; Freire, C., Progress in the Raman spectra analysis of covalently functionalized multiwalled carbon nanotubes: unraveling disorder in graphitic materials Phys. Chem. Chem. Phys. 2016, 18, 12784.