Publications 2016

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Strub, D.J.; Salat, K.; Librowski, T.; Lochynski, S.; Gawel, M.; Podkowa, A., The anxiolytic-like activity of a novel N-cycloalkyl- N-benzoylpiperazine derivative. Pharm. Rep. 2016, 68, 62.

Kosikowska, P.; Bochno, M.; Macegoniuk, K.; Forlani, G.; Kafarski, P.; Berlicki, Ł., Bisphosphonic acids as effective inhibitors of Mycobacterium tuberculosis glutamine synthetase J. Enz. Inh. Med. Chem. 2016, 31, 931.

Strub, D.J.; Kula, J.; Sikora, M.; Gibka, J.; Lochynski, S., Synthesis and olfactory evaluation of homologous series of (+)- and (-)-carvone oxime ethers Flavour Frag. J. 2016, 31, 81.

Gersch M, Stahl M, Poreba M, Dahmen M, Dziedzic A, Drag M, Sieber SA, Barrel-shaped ClpP proteases display attenuated cleavage specificity ACS Chemical Biology 2016, 11, 389.

Ząbek, A.; Swierkot, J; Malak, A.; Zawadzka, I.; Deja, S.; Bogunia-Kubik, K.; Mlynarz, P. , Application of H-1 NMR-based serum metabolomic studies for monitoring female patients with rheumatoid arthritis J. Pharm. Biomed. Anal. 2016, 117, 544.

Wójcik, P.; Berlicki, Ł., Peptide-based inhibitors of protein–protein interactions. Bioorg. Med. Chem. Lett. 2016, 26, 707.

Byzia, A.; Szeffler, A.; Kalinowski, L.; Drąg, M., Activity profiling of aminopeptidases in cell lysates using a fluorogenic substrate library Biochimie 2016, 122, 31.

Górny vel Górniak, M.; Kafarski, P., Preparation of the library of fluorescent aromatic aminophosphonate phenyl and benzyl esters Phosphorus, Sulfur, Silicon Relat. Elem. 2016, 191, 511.

Wysoczański, T., Sokoła-Wysoczańska, E., Pękala, J., Lochyński, S., Czyż K., Bodkowski, R., Herbinger, G., Patkowska-Sokoła, B., Librowski, T., Omega-3 Fatty Acids and their Role in Central Nervous System - A Review Curr. Med. Chem. 2016, 23, 816.

Modak, J. K.; Rut, W.; Wijeyewickrema, L. C.; Pike, R. N.; Drąg, M.; Roujeinkova, A., Structural basis for substrate specificity of Helicobacter pylori M17 aminopeptidase Biochimie 2016, 121, 60.

Węglarz-Tomczak, E.; Berlicki, Ł.; Pawełczak, M.; Nocek, B.; Joachimiak, A. Mucha, A., A structural insight into the P1-S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases. Eur. J. Med. Chem. 2016, 117, 187.

Orczyk-Pawiłowicz, M.; Jawień, E.; Deja, S.; Hirnle, L.; Ząbek, A.; Młynarz, P., Metabolomics of Human Amniotic Fluid and Maternal Plasma furing Normal Pregnancy PLoS One 2016, 11, 1.

Majewska, P.; Serafin, M., Klimek-Ochab, M.; Brzezińska-Rodak, M.; Żymańczyk-Duda, E., Lipases and whole cell biotransformations of 2-hydroxy-2-(ethoxyphenylphosphinyl)acetic acid and its ester Bioorg. Chem. 2016, 66, 21.

Brzezińska-Rodak, M.; Klimek-Ochab, M.; Żymańczyk-Duda, E., Enzyme-mediated protoplast formation of Cuninghamella echinulata – preliminary studies BioTechnologia 2016, 97, 27.

Chmielewska, E.; Kafarski, P., Physiologic Activity of Bisphosphonates – Recent Advances Open Pharm. Sci. J. 2016, 3, 56.

Dziuganowska, Z. A.; Ślepokura, A.; Volle, J.-N.; Virieux, D.; Pirat, J.-L.; Kafarski, P., Structural Analogues of Selfotel J. Org. Chem. 2016, 81, 4947.

Deiasna, M.; Pokładek, Z.; Olesiak-Bańska, J.; Młynarz, P.; Samoć, M.; Matczyszyn., K., Photochromic switching of the DNA helicity induced by azobenzene derivatives Sci. Rep. 2016, 6, 1.

Macegoniuk, K.; Grela, E.; Palus, J.; Rudzińska-Szostak, E.; Grabowiecka, A.; Biernat, M.; Berlicki, Ł., 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. J. Med. Chem. 2016, 59, 8125.

Węglarz-Tomczak, E.; Vassiliou, S.; Mucha, A., Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues. Bioorg. Med. Chem. Lett. 2016, 26, 4122.

Węglarz-Tomczak, E.; Staszewska, K.; Talma, M.; Mucha, A., Enantiomeric a,ß-diaminoethylphosphonic acids as potent inhibitors of aminopeptidases — stereoselective synthesis and biological activity. Tetrahedron Lett. 2016, 57, 4812.

Węglarz-Tomczak, E.; Burda-Grabowska, M.; Giurg, M.; Mucha, A., Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study. Bioorg. Med. Chem. Lett. 2016, 26, 5254.

Górak, M.; Żymańczyk-Duda, E., Reductive activity of free and immobilized cells of cyanobacteria toward oxophosphonates—comparative study J. Appl. Phycol. 2016, 1.

Rut, W.; Drąg, M., Human 20S proteasome activity towards fluorogenic peptides of various chain lengths Biol. Chem. 2016, 396, 921.

Grela, E.; Dziełak, A.; Szydowska, K.; Mucha, A.; Kafarski, P.; Grabowiecka, A.M., Whole-cell Proteus mirabilis urease inhibition by aminophosphinates for the control of struvite formation. J. Med. Microbiol. 2016, 65, 1123.

Chmielewska, E.; Kafarski, P., Synthetic procedures leading towards aminobisphosphonates Molecules 2016, 21, 1.

Dobosz, A.; Spychała, J.; Ptak, T.; Chmielewska, E.; Maciejewska, G.; Kafarski, P.; Młynarz, P. , Electrochemical and spectroscopic investigations of selected N-heteroalkylaminomethylenebisphosphonic acids with Pb(II) ions Coord. Chem. Rev. 2016, 327-328, 271.

Drinkwater N, Sivaraman KK, Bamert RS, Rut W, Mohamed K, Vinh NB, Scammells PJ, Drag M, McGowan S, Structure and substrate fingerprint of aminopeptidase P from Plasmodium falciparum Biochemical Journal 2016, 473, 3189.

Poreba M, Solberg R, Rut W, Lunde NN, Kasperkiewicz P, Snipas SJ, Mihelic M, Turk D, Turk B, Salvesen GS, Drag M., Counter Selection Substrate Library Strategy for Developing Specific Protease Substrates and Probes Cell Chemical Biology 2016, 23, 1023.

Lentz CS, Ordonez AA, Kasperkiewicz P, La Greca F, O'Donoghue AJ, Schulze CJ, Powers JC, Craik CS, Drag M, Jain SK, Bogyo M, Design of Selective Substrates and Activity-Based Probes for Hydrolase Important for Pathogenesis 1 (HIP1) from Mycobacterium tuberculosis. ACS infectious diseases 2016, 2, 807.

Majewska P, Serafin M, Klimek-Ochab M, Brzezińska-Rodak M, Żymańczyk-Duda E,, Lipases and whole cell biotransformations of 2-hydroxy-2-(ethoxyphenylphosphinyl)acetic acid and its ester. Bioorganic Chemistry 2016, 66, 21.

Brzezińska-Rodak M, Klimek-Ochab M, Żymańczyk-Duda E, Enzyme-mediated protoplast formation of Cuninghamella echinulata - preliminary studies. BioTechnologia 2016, 97, 27.

Jewginski, M., Fischer, L., Colombo, C., Huc, I., MacKereth, C.D., Solution Observation of Dimerization and Helix Handedness Induction in a Human Carbonic Anhydrase-Helical Aromatic Amide Foldamer Complex ChemBioChem 2016, 17, 727.

Lamch Ł., Tylus W., Jewgiński M., Latajka R., Wilk K.A., Location of Varying Hydrophobicity Zinc(II) Phthalocyanine-Type Photosensitizers in Methoxy Poly(ethylene oxide) and Poly(l-lactide) Block Copolymer Micelles Using 1H NMR and XPS Techniques J. Phys. Chem. B 2016, 120, 12768–12780.

Żymańczyk-Duda E, Brzezińska-Rodak M, Klimek-Ochab M, Duda M, Biochemistry - Knowledge to Practical Applications - Examples Basic Biochemistry 2016, 1.