Publications 2020

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Hałdys K., Goldeman W., Jewgiński M., Wolińska E., Anger-Góra N., Rossowska J., Latajka R., Halogenated aromatic thiosemicarbazones as potent inhibitors of tyrosinase and melanogenesis Bioorganic Chemistry 2020, 94, 103419.

Mucha, A.; Kafarski, P., Peptide and Pseudopeptide Bond Synthesis in Phosphorus Dipeptide Analogs. Methods Mol. Biol. 2020, 2103, 287.

Petruczynik, P.; Kafarski, P.; Psurski, M.; Wietrzyk, J.; Kiełbowicz, Z.; Kuryszko, J.; Chmielewska, E. , Three-Component Reaction od Diamines with Triethyl Orthoformate and Diethyl Phosphite and Anti-Proliferative and Antiosteoporotic Activities of the Products Molecules 2020, 25, 1.

Wanat, W.; Talma, M.; Dziuk, B.; Pirat, J.-L.; Kafarski, P., Phosphonic Acid Analogs of Fluorophenylalanines as Inhibitors of Human and Porcine Aminopeptidases N: Validation of the Importance of the Substitution of the Aromatic Ring Biomolecules 2020, 10, 1.

Wanat, W.; Dziuk, B.; Kafarski, P., New crystal structures of fluorinated α-aminophosphonic acid analogues of phenylglycine Struct. Chem. 2020, 31, 1197.

Talma, M.; Mucha, A., P1′ Residue-Oriented Virtual Screening for Potent and Selective Phosphinic (Dehydro) Dipeptide Inhibitors of Metallo-Aminopeptidases Biomolecules 2020, 10, 659.

Lenartowicz, P.; Witkowska, D.; Żyszka-Haberecht, B.; Dziuk, B.; Ejsmont, K.; Świątek-Kozłowska, J.; Kafarski, P., A novel approach for obtaining alpha,beta-diaminophosphonates bearing structurally diverseside chains and their interactions with transition metal ions studied by ITC RSC Adv. 2020, 10, 24045.

Tarczewska, A.; Wycisk, K.; Orłowski, M.;Waligórska, A.; Dobrucki, J.; Drewniak-Świtalska, M.; Berlicki, Ł.; Ożyhar, A., Nuclear immunophilin FKBP39 from Drosophila melanogaster drives spontaneous liquid-liquid phase separation. Int. J. Biol. Macromol. 2020, 163, 108.

Kafarski, P., Phosphonopeptides containing free phosphonic groups: recent advances RCS Adv. 2020, 10, 25898.

Fortuna, P.; Linhares, B. M.; Purohit, T.; Pollock, J.; Cierpicki, T.; Grembecka, J.; Berlicki, Ł., Covalent and noncovalent constraints yield a figure eight-like conformation of a peptide inhibiting the menin-MLL interaction Eur. J. Med. Chem. 2020, 207, 112748.

Wanat, W. ; Talma, M.; Dziuk, B.; Kafarski, P, Synthesis and Inhibitory Studies of Phosphonic Acid Analogues of Homophenylalanine and Phenylalanine towards Alanyl Aminopeptidases Biomolecules 2020, 10, 1.

Fortuna, P.; Twarda-Clapa, A.; Skalniak, L.; Ożga, K.; Holak, T. A.; Berlicki, Ł., Systematic ‘foldamerization’ of peptide inhibiting p53-MDM2/X interactions by the incorporation of trans- or cis-2-aminocyclopentanecarboxylic acid residues Eur. J. Med. Chem. 2020, 208, 112814.

Janiszewska, K.; Talma, M.; Oszywa, B.; Pawełczak, M.; Kafarski, P.; Mucha, A.,, N-Benzyl Residues as the P1' Substituents in Phosphorus-Containing Extended Transition State Analog Inhibitors of Metalloaminopeptidases Molecules 2020, 25, 4334.

Errante F.; Ledwoń P.; Latajka R.; Rovero P.; Papini A.M., Cosmeceutical Peptides in the Framework of Sustainable Wellness Economy Frontiers in Chemistry 2020, 8, 572923.

Fernández-Pérez, H.; Lenartowicz, P.; Carreras, L.; Grabulosa, A.; Kafarski, P.; Vidal-Ferran, A., Access to α-Aminophosphonic Acid Derivatives and Phosphonopeptides by [Rh(P–OP)]-Catalyzed Stereoselective Hydrogenation J. Org. Chem. 2020, 85, 14779.

Dajek, M.; Pruszczyńska, A.; Konieczny, K. A.; Kowalczyk, R., Cinchona squaramide-catalyzed intermolecular desymmetrization of 1,3-diketones leading to chiral 1,4-dihydropyridines. Adv. Synth. Catal. 2020, 362, 3613.