Publications 2020

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Hałdys K., Goldeman W., Jewgiński M., Wolińska E., Anger-Góra N., Rossowska J., Latajka R., Halogenated aromatic thiosemicarbazones as potent inhibitors of tyrosinase and melanogenesis Bioorganic Chemistry 2020, 94, 103419.

Mucha, A.; Kafarski, P., Peptide and Pseudopeptide Bond Synthesis in Phosphorus Dipeptide Analogs. Methods Mol. Biol. 2020, 2103, 287.

Rut W, Groborz K, Zhang L, Modrzycka S, Poreba M, Hilgenfeld R, Drag M, Profiling of flaviviral NS2B-NS3 protease specificity provides a structural basis for the development of selective chemical tools that differentiate dengue from Zika and West Nile viruses Antiviral Research 2020, 1.

Poreba M, Protease-activated prodrugs: strategies, challenges and future directions FEBS Journal 2020, 1.

Rut W, Groborz K, Zhang L, Sun X, Zmudzinski M, Hilgenfeld R, Drag M, Substrate specificity profiling of SARS-CoV-2 Mpro protease provides basis for anti-COVID-19 drug design bioRxiv 2020, 1.

Rut W, Żmudziński M, Snipas SJ, Bekes M, Huang TT, Drag M, Engineered unnatural ubiquitin for optimal detection of deubiquitinating enzymes Chemical Science 2020, 1.

Petruczynik, P.; Kafarski, P.; Psurski, M.; Wietrzyk, J.; Kiełbowicz, Z.; Kuryszko, J.; Chmielewska, E. , Three-Component Reaction od Diamines with Triethyl Orthoformate and Diethyl Phosphite and Anti-Proliferative and Antiosteoporotic Activities of the Products Molecules 2020, 25, 1.

Aaltonen N, Singha PK, Jakupović H, Wirth T, Samaranayake H, Pasonen-Seppänen S, Rilla K, Varjosalo M, Edgington-Mitchell LE, Kasperkiewicz P, Drag M, Kälvälä S, Moisio E, Savinainen JR, Laitinen JT, High-Resolution Confocal Fluorescence Imaging of Serine Hydrolase Activity in Cryosections - Application to Glioma Brain Unveils Activity Hotspots Originating from Tumor-Associated Neutrophils. Biological Procedures Online 2020, 22, 1.

Kołt S, Janiszewski T, Kaiserman D, Modrzycka S, Snipas SJ, Salvesen G, Dra G M, Bird PI, Kasperkiewicz P, Detection of Active Granzyme A in NK92 Cells with Fluorescent Activity-Based Probe. Journal of Medicinal Chemistry 2020, 1.

Wanat, W.; Talma, M.; Dziuk, B.; Pirat, J.-L.; Kafarski, P., Phosphonic Acid Analogs of Fluorophenylalanines as Inhibitors of Human and Porcine Aminopeptidases N: Validation of the Importance of the Substitution of the Aromatic Ring Biomolecules 2020, 10, 1.

Wanat, W.; Dziuk, B.; Kafarski, P., New crystal structures of fluorinated α-aminophosphonic acid analogues of phenylglycine Struct. Chem. 2020, 31, 1197.

Talma, M.; Mucha, A., P1′ Residue-Oriented Virtual Screening for Potent and Selective Phosphinic (Dehydro) Dipeptide Inhibitors of Metallo-Aminopeptidases Biomolecules 2020, 10, 659.

Maniak, H.; Talma, M.; Matyja, K.; Trusek, A.; Giurg, M. , Synthesis and structure-activity relationship studies of hydrazide-hydrazones as inhibitors of laccase from trametes versicolor Molecules 2020, 5, 1255.

Talma, M., Phosphinic Dehydrodipeptides: Diversification of the P1′ Residue with the Morita–Baylis–Hillman Acetates and Inhibition of Alanyl Aminopeptidase Int J Pept Res Ther 2020, 1.

Lenartowicz, P.; Witkowska, D.; Żyszka-Haberecht, B.; Dziuk, B.; Ejsmont, K.; Świątek-Kozłowska, J.; Kafarski, P., A novel approach for obtaining alpha,beta-diaminophosphonates bearing structurally diverseside chains and their interactions with transition metal ions studied by ITC RSC Advances 2020, 10, 24045.

Janiszewski T, Kolt S, Kaiserman D, Snipas SJ, Li S, Kulbacka J, Saczko J, Bovenschen N, Salvesen G, Drag M, Bird P, Kasperkiewicz P, Noninvasive optical detection of granzyme B from natural killer cells with enzyme-activated fluorogenic probes Journal of Biological Chemistry 2020, 1.

Bibo-Verdugo B, Snipas SJ, Kolt S, Poreba M, Salvesen GS, Extended subsite profiling of the pyroptosis effector protein gasdermin D reveals a region recognized by inflammatory caspase-11 Journal of Biological Chemistry 2020, 1.

Tholen M, Yim JJ, Groborz K, Yoo E, Martin BA, van der Berg NS, Drag M, Bogyo M, Design of optical imaging probes by screening of diverse substrate libraries directly in disease tissue extracts Angewandte Chemie 2020, 1.

Skowron PM, Krefft D, Brodzik R, Kasperkiewicz P, Drag M, Koller KP, An Alternative for Proteinase K-heat-sensitive Protease From Fungus Onygena Corvina for Biotechnology: Cloning, Engineering, Expression, Characterization and Special Application for Protein Sequencing Microbial Cell Factories 2020, 19, 135.

Tarczewska, A.; Wycisk, K.; Orłowski, M.;Waligórska, A.; Dobrucki, J.; Drewniak-Świtalska, M.; Berlicki, Ł.; Ożyhar, A., Nuclear immunophilin FKBP39 from Drosophila melanogaster drives spontaneous liquid-liquid phase separation. Int. J. Biol. Macromol. 2020, 163, 108.

Razai AS, Snipas SJ, Poreba M, Fasci D, Salvesen GS, Engineering Caspase 7 as an Affinity Reagent to Capture Proteolytic Products The FEBS Journal 2020, 1.

Kafarski, P., Phosphonopeptides containing free phosphonic groups: recent advances ACS Adv. 2020, 10, 25898.